Olanzapine effects on body composition, food preference, glucose metabolism and insulin sensitivity in the rat

Arch Physiol Biochem. 2011 Oct;117(4):241-9. doi: 10.3109/13813455.2011.576681. Epub 2011 Jun 15.

Abstract

The atypical antipsychotic drug olanzapine induces weight gain and defects in glucose metabolism in patients. Using a rat model we investigated the effects of acute and long term olanzapine treatment on weight gain, food preference and glucose metabolism. Olanzapine treated rats fed a chow diet grew more slowly than vehicle controls but olanzapine treated animals fed a high fat/sugar diet grew faster than control animals on the same diet. These changes in weight were paralleled by changes in fat mass. Olanzapine also induced a strong preference for a high fat/high sugar diet. Acute exposure to olanzapine rapidly induced severe impairments of glucose tolerance and increased insulin secretion but did not impair insulin tolerance. These results indicate the defect in glucose metabolism induced by acute olanzapine treatment was most likely due to increased hepatic glucose output associated with a reduction in active GLP-1 levels and correspondingly high glucagon levels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antipsychotic Agents / adverse effects
  • Antipsychotic Agents / pharmacology*
  • Antipsychotic Agents / therapeutic use
  • Benzodiazepines / adverse effects
  • Benzodiazepines / pharmacology*
  • Benzodiazepines / therapeutic use
  • Body Composition / drug effects*
  • Body Weight / drug effects
  • Diet, High-Fat / adverse effects
  • Diet, High-Fat / psychology
  • Food Preferences / drug effects*
  • Food Preferences / psychology
  • Glucagon / metabolism
  • Glucagon-Like Peptide 1 / antagonists & inhibitors
  • Glucagon-Like Peptide 1 / biosynthesis
  • Glucose / metabolism*
  • Glucose Tolerance Test
  • Humans
  • Insulin / metabolism*
  • Insulin Resistance*
  • Liver / drug effects*
  • Liver / metabolism
  • Male
  • Obesity / metabolism
  • Olanzapine
  • Rats
  • Schizophrenia / drug therapy
  • Weight Gain / drug effects

Substances

  • Antipsychotic Agents
  • Insulin
  • Benzodiazepines
  • Glucagon-Like Peptide 1
  • Glucagon
  • Glucose
  • Olanzapine