Is high-dose nafamostat mesilate effective for the prevention of post-ERCP pancreatitis, especially in high-risk patients?

Pancreas. 2011 Nov;40(8):1215-9. doi: 10.1097/MPA.0b013e31822116d5.

Abstract

Objective: Infusion of the protease inhibitor nafamostat mesilate (20 mg) effectively prevents post-ERCP pancreatitis, but only in low-risk groups. This study was performed to evaluate the use of high-dose nafamostat mesilate (50 mg) for prevention of post-ERCP pancreatitis (PEP), especially in high-risk groups.

Methods: A total of 608 patients who underwent ERCP were included; 13 patients were excluded. Patients were divided into 3 groups: controls (group A), infusion with 20 mg of nafamostat mesilate (group B), or infusion with 50 mg of nafamostat mesilate (group C). The incidence of PEP was analyzed.

Results: The overall incidence of acute pancreatitis was 7.4% (44/595). There was a significant difference in the incidence of PEP with or without nafamostat mesilate (13.0% vs 4.0% and 5.1%, respectively; P < 0.0001). Subgroup analysis showed that in low-risk patients, the rate of PEP was significantly different with nafamostat (11.9% vs 2.7% and 4.0%, respectively; P = 0.007). In high-risk patients, the rate of PEP was not significantly different among treatment groups (14.6% vs 5.9% vs 6.9%, respectively; P = 0.108).

Conclusions: Nafamostat mesilate prophylaxis (20 or 50 mg) is effective in preventing post-ERCP pancreatitis. However, the preventive effect of high-dose nafamostat mesilate (50 mg) is not significant in high-risk patients.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute Disease
  • Aged
  • Amylases / blood
  • Benzamidines
  • Cholangiopancreatography, Endoscopic Retrograde / adverse effects*
  • Dose-Response Relationship, Drug
  • Drug Administration Schedule
  • Female
  • Guanidines / administration & dosage
  • Guanidines / therapeutic use*
  • Humans
  • Infusions, Intravenous
  • Male
  • Middle Aged
  • Pancreatitis / blood
  • Pancreatitis / etiology
  • Pancreatitis / prevention & control*
  • Prospective Studies
  • Protease Inhibitors / administration & dosage
  • Protease Inhibitors / therapeutic use
  • Risk Factors
  • Time Factors
  • Treatment Outcome

Substances

  • Benzamidines
  • Guanidines
  • Protease Inhibitors
  • Amylases
  • nafamostat