Evaluation of effects of low-dose aspirin administration on urinary thromboxane metabolites in healthy dogs

Am J Vet Res. 2011 Aug;72(8):1038-45. doi: 10.2460/ajvr.72.8.1038.

Abstract

Objective: To evaluate markers of in vivo platelet function (urinary 11-dehydro-thromboxane B(2) [11-dehydroTXB(2)] and 2,3-dinorTXB(2)) and assess their response to administration of 2 commonly used dosages of aspirin in healthy dogs.

Animals: 20 healthy dogs.

Procedures: Urine was collected prior to aspirin administration and on the morning following the last evening administration. Twenty dogs received aspirin (1 mg/kg, PO, q 24 h) for 7 consecutive doses. After a washout period of 5 months, 10 dogs received a single dose of aspirin (10 mg/kg, PO). Concentrations of urinary thromboxane metabolites 11-dehydroTXB(2) and 2,3-dinorTXB(2) were measured via ELISA, and values were normalized to urine creatinine concentration.

Results: Median baseline 11-dehydroTXB(2) concentrations were 0.38 ng/mg of creatinine (range, 0.15 to 1.13 ng/mg). Mean ± SD baseline 2 at a 3-dinorTXB(2) concentrations were 6.75 ± 2.77 ng/mg of creatinine. Administration of aspirin at a dosage of 1 mg/kg, PO, every 24 hours for 7 days did not significantly decrease urinary 11-dehydroTXB(2) concentration, but administration of the single aspirin dose of 10 mg/kg did significantly decrease 11-dehydroTXB(2) concentration by a median of 45.5% (range, 28.2% to 671%). Administration of the 1 mg/kg aspirin dosage significantly decreased urinary 2,3-dinorTXB(2) concentration by a mean ± SD of 33.0 ± 23.7%. Administration of the single aspirin dose of 10 mg/kg also significantly decreased 2,3-dinorTXB(2) concentration by a mean ± SD of 46.7 ± 12.6%.

Conclusions and clinical relevance: Aspirin administration (1 mg/kg/d) may be insufficient for reliable platelet inhibition in healthy dogs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Aspirin / administration & dosage
  • Aspirin / pharmacology*
  • Dogs / physiology*
  • Enzyme-Linked Immunosorbent Assay / veterinary
  • Female
  • Male
  • Platelet Aggregation Inhibitors / administration & dosage
  • Platelet Aggregation Inhibitors / pharmacology*
  • Thromboxane B2 / analogs & derivatives
  • Thromboxane B2 / metabolism
  • Thromboxane B2 / urine

Substances

  • Platelet Aggregation Inhibitors
  • Thromboxane B2
  • 2,3-dinor-thromboxane B2
  • 11-dehydro-thromboxane B2
  • Aspirin