Structure of N5-carboxyaminoimidazole ribonucleotide synthase (PurK) from Bacillus anthracis

Acta Crystallogr D Biol Crystallogr. 2011 Oct;67(Pt 10):870-4. doi: 10.1107/S0907444911029210. Epub 2011 Sep 8.

Abstract

The apo structure of N5-carboxyaminoimidazole ribonucleotide synthase (PurK) from Bacillus anthracis (baPurK) with Mg2+ in the active site is reported at 1.96 Å resolution. PurK is an enzyme in the purine-biosynthetic pathway, unique to prokaryotes, that converts 5-aminoimidazole ribonucleotide to N5-carboxyaminoimidazole ribonucleotide and has been suggested as a potential antimicrobial drug target. Two interesting features of baPurK are a flexible B-loop (residues 149/150-157) that is in close contact with the active site and the binding of Mg2+ to the active site without additional ligands.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Bacillus anthracis / enzymology*
  • Bacterial Proteins / chemistry
  • Binding Sites
  • Catalytic Domain
  • Crystallography, X-Ray
  • Imidazoles / metabolism
  • Ligases / chemistry*
  • Ligases / metabolism
  • Magnesium / metabolism
  • Protein Conformation

Substances

  • Bacterial Proteins
  • Imidazoles
  • 4-aminoimidazole
  • Ligases
  • Magnesium

Associated data

  • PDB/3Q2O