Domino reactions for the synthesis of various α-substituted nitro alkenes

Org Biomol Chem. 2012 Jan 21;10(3):524-8. doi: 10.1039/c1ob06260c. Epub 2011 Oct 24.

Abstract

Efficient one-pot methods for the synthesis of variously functionalised conjugated nitro alkenes have been reported. Despite the utility in different fields of these compounds, only a few multi-step syntheses have been reported in the literature, giving the target compounds in low overall yields. α-Nitro acrylates or cinnamates, α-nitro α,β-unsaturated ketones and, most importantly, aromatic and heteroaromatic (E)- 2-nitro allylic alcohols, compounds characterised by a well-known anticancer activity, were obtained in high yields and high diastereomeric purity by a domino condensation-dehydration process.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkenes / chemical synthesis*
  • Alkenes / chemistry*
  • Chemistry Techniques, Synthetic / methods*
  • Nitro Compounds / chemical synthesis*
  • Nitro Compounds / chemistry*
  • Stereoisomerism
  • Substrate Specificity

Substances

  • Alkenes
  • Nitro Compounds