[Synthesis and spectral characteristic of pharmaceutical dipfluzine hydrochloride-benzoic acid co-crystal]

Guang Pu Xue Yu Guang Pu Fen Xi. 2011 Sep;31(9):2476-9.
[Article in Chinese]

Abstract

Pharmaceutical co-crystals can improve the chemical and physical properties of active pharmaceutical ingredient (API), which is new idea and expected to provide new stable structures. Pharmaceutical co-crystals have the potential to be much more useful in pharmaceutical products than salts, solvates or hydrates, polymorphs and stoichiometric solvates (pseudo-polymorphs). In our study, dipfluzine hydrochloride-benzoic acid co-crystal was synthesized by solid co-grinding. The samples were subjected to IR, DSC, XRD, Raman and THz spectral analysis. The results indicated that dipfluzine hydrochloride-benzoic acid complex was new phase compared with the single API and CCF. THz-TDS characterization indicated that hydrogen bond formed between API and CCF, which confirmed the formation of co-crystal.

MeSH terms

  • Benzoic Acid*
  • Cinnarizine / analogs & derivatives*
  • Cinnarizine / chemical synthesis
  • Cinnarizine / chemistry
  • Crystallization
  • Hydrogen Bonding
  • Spectrum Analysis

Substances

  • Cinnarizine
  • dipfluzine
  • Benzoic Acid