Abstract
The presenilin complex is composed of four core proteins (presenilin 1 or presenilin 2, APH1, nicastrin, and PEN2). Several endogenous proteins have been reported to selectively modulate the function of the presenilin complexes; these include transmembrane trafficking protein, 21-KD (TMP21), CD147 antigen (basigin), the γ-secretase-activating protein (gSAP), and the orphan G-protein-coupled receptor 3. Because the structure and assembly of these complexes underlies their activity, this review will discuss current work on the assembly of the complex and on presenilin-interacting proteins that regulate secretase activity.
© 2011 The Authors. Journal of Neurochemistry © 2011 International Society for Neurochemistry.
MeSH terms
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Alzheimer Disease / enzymology*
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Alzheimer Disease / metabolism
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Amyloid Precursor Protein Secretases / chemistry
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Amyloid Precursor Protein Secretases / metabolism*
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Amyloid Precursor Protein Secretases / physiology
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Amyloid beta-Peptides / chemistry
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Amyloid beta-Peptides / metabolism
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Animals
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Endopeptidases
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Humans
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Membrane Proteins / chemistry
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Membrane Proteins / physiology
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Peptide Hydrolases / chemistry
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Peptide Hydrolases / physiology
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Presenilin-1 / chemistry*
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Presenilin-1 / physiology
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Presenilin-2 / chemistry*
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Presenilin-2 / physiology
Substances
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Amyloid beta-Peptides
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Membrane Proteins
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PSEN1 protein, human
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PSENEN protein, human
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Presenilin-1
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Presenilin-2
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APH1A protein, human
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Amyloid Precursor Protein Secretases
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Endopeptidases
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Peptide Hydrolases