Abstract
The search for safe, non-addictive versions of morphine and other opioid drugs has just received a boost with the solving of the crystal structures of the receptors to which the drugs bind.
MeSH terms
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Animals
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Biomimetic Materials / chemistry*
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Humans
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Morphinans / chemistry*
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Naltrexone / analogs & derivatives*
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Naltrexone / chemistry
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Opioid Peptides / chemistry*
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Piperidines / chemistry*
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Piperidines / metabolism*
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Receptors, Opioid / chemistry*
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Receptors, Opioid / metabolism*
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Receptors, Opioid, delta / chemistry*
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Receptors, Opioid, kappa / antagonists & inhibitors*
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Receptors, Opioid, kappa / chemistry*
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Receptors, Opioid, mu / antagonists & inhibitors*
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Receptors, Opioid, mu / chemistry*
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Spiro Compounds / chemistry*
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Spiro Compounds / metabolism*
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Tetrahydroisoquinolines / chemistry*
Substances
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(Nphe(1),Arg(14),Lys(15))N-OFQ NH(2)
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1-benzyl-N-(3-(spiroisobenzofuran-1(3H),4'-piperidin-1-yl)propyl)pyrrolidine-2-carboxamide
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7-hydroxy-N-(1-((4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl)methyl)-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide
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Morphinans
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Opioid Peptides
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Piperidines
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Receptors, Opioid
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Receptors, Opioid, delta
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Receptors, Opioid, kappa
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Receptors, Opioid, mu
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Spiro Compounds
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Tetrahydroisoquinolines
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Naltrexone
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nociceptin receptor
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naltrindole