In vitro and in vivo kinetic analysis of the interaction of a norbornyl derivative of propranolol with beta-adrenergic receptors of brain and C6 glioma cells; an irreversible or slowly reversible ligand

Mol Pharmacol. 1979 May;15(3):588-97.
No abstract available

MeSH terms

  • Adenylyl Cyclase Inhibitors
  • Animals
  • Binding, Competitive
  • Brain / metabolism*
  • Bridged Bicyclo Compounds / metabolism
  • Cells, Cultured
  • Dihydroalprenolol / metabolism
  • Glioma / metabolism*
  • In Vitro Techniques
  • Kinetics
  • Ligands
  • Male
  • Neoplasms, Experimental / metabolism
  • Propanolamines / metabolism*
  • Rats
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, beta / metabolism*

Substances

  • Adenylyl Cyclase Inhibitors
  • Bridged Bicyclo Compounds
  • Ligands
  • Propanolamines
  • Receptors, Adrenergic
  • Receptors, Adrenergic, beta
  • Dihydroalprenolol