Iron(III)-doped, silica nanoshells: a biodegradable form of silica

J Am Chem Soc. 2012 Aug 29;134(34):13997-4003. doi: 10.1021/ja3036114. Epub 2012 Aug 16.

Abstract

Silica nanoparticles are being investigated for a number of medical applications; however, their use in vivo has been questioned because of the potential for bioaccumulation. To obviate this problem, silica nanoshells were tested for enhanced biodegradability by doping iron(III) into the nanoshells. Exposure of the doped silica to small molecule chelators and mammalian serum was explored to test whether the removal of iron(III) from the silica nanoshell structure would facilitate its degradation. Iron chelators, such as EDTA, desferrioxamine, and deferiprone, were found to cause the nanoshells to degrade on the removal of iron(III) within several days at 80 °C. When the iron(III)-doped, silica nanoshells were submerged in fetal bovine and human serums at physiological temperature, they also degrade via removal of the iron by serum proteins, such as transferrin, over a period of several weeks.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Biocompatible Materials / chemistry*
  • Biocompatible Materials / metabolism
  • Cattle
  • Deferiprone
  • Deferoxamine / metabolism
  • Edetic Acid / metabolism
  • Ferric Compounds / chemistry*
  • Ferric Compounds / metabolism
  • Humans
  • Iron Chelating Agents / metabolism
  • Nanoshells / chemistry*
  • Nanoshells / ultrastructure
  • Pyridones / metabolism
  • Serum / metabolism
  • Silicon Dioxide / chemistry*
  • Silicon Dioxide / metabolism
  • Transferrin / metabolism

Substances

  • Biocompatible Materials
  • Ferric Compounds
  • Iron Chelating Agents
  • Pyridones
  • Transferrin
  • Deferiprone
  • Silicon Dioxide
  • Edetic Acid
  • Deferoxamine