Use of metabolite AUC data in bioavailability studies to discriminate between absorption and first-pass extraction

Clin Pharmacokinet. 1990 May;18(5):419-22. doi: 10.2165/00003088-199018050-00006.
No abstract available

MeSH terms

  • Absorption
  • Antipyrine / pharmacokinetics
  • Biological Availability*
  • Caffeine / pharmacokinetics
  • Diphenhydramine / pharmacokinetics
  • Dose-Response Relationship, Drug*
  • Humans
  • Ketanserin / pharmacokinetics
  • Lidocaine / pharmacokinetics
  • Liver Diseases / metabolism
  • Metronidazole / pharmacokinetics
  • Nomifensine / pharmacokinetics
  • Triamterene / pharmacokinetics

Substances

  • Metronidazole
  • Nomifensine
  • Caffeine
  • Diphenhydramine
  • Ketanserin
  • Lidocaine
  • Antipyrine
  • Triamterene