Mechanistic basis of phenothiazine-driven inhibition of Tau aggregation

Angew Chem Int Ed Engl. 2013 Mar 18;52(12):3511-5. doi: 10.1002/anie.201208290. Epub 2013 Feb 11.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alzheimer Disease / metabolism
  • Alzheimer Disease / pathology
  • Animals
  • Caenorhabditis elegans / drug effects
  • Caenorhabditis elegans / metabolism
  • Cysteine / chemistry
  • Disease Models, Animal
  • Humans
  • Magnetic Resonance Spectroscopy
  • Methylene Blue / chemistry
  • Oxidation-Reduction
  • Phenothiazines / chemistry*
  • Phenothiazines / metabolism
  • Phenothiazines / pharmacology
  • Protein Binding
  • tau Proteins / antagonists & inhibitors*
  • tau Proteins / metabolism

Substances

  • Phenothiazines
  • tau Proteins
  • phenothiazine
  • Cysteine
  • Methylene Blue