Dissociation kinetics of a binary complex in solution by protein displacement

Angew Chem Int Ed Engl. 2013 Nov 25;52(48):12587-91. doi: 10.1002/anie.201306253. Epub 2013 Oct 7.
No abstract available

Keywords: NMR spectroscopy; kinetics; ligand-protein complexes; off-rate constants; proteins.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cyclophilin A / chemistry
  • Cyclophilin A / metabolism*
  • Cyclosporine / chemistry
  • Cyclosporine / metabolism*
  • Immunosuppressive Agents / chemistry
  • Immunosuppressive Agents / metabolism*
  • Kinetics
  • Ligands
  • Models, Molecular
  • Nuclear Magnetic Resonance, Biomolecular

Substances

  • Immunosuppressive Agents
  • Ligands
  • Cyclosporine
  • Cyclophilin A
  • alisporivir