Age-dependent increase in [3H]verapamil binding to rat cortical membranes

Neurosci Lett. 1985 Oct 24;61(1-2):67-71. doi: 10.1016/0304-3940(85)90402-1.

Abstract

[3H]Nitrendipine bound to cerebral cortex membranes is displaced more efficiently by verapamil in old rats (24 months old) compared to young ones (3 months old). In addition, [3H]verapamil binding was studied in detail in 3-, 12- and 24-month-old rats. Aging increases the Bmax of [3H]verapamil, leaving the affinity unchanged. These observations further indicate that aging may affect calcium channels leading to a derangement of calcium movements which in turn alter neuronal activity.

Publication types

  • Comparative Study

MeSH terms

  • Age Factors
  • Aging*
  • Animals
  • Binding, Competitive
  • Calcium / metabolism*
  • Cerebral Cortex / metabolism*
  • Ion Channels / metabolism*
  • Male
  • Membranes / metabolism
  • Nifedipine / analogs & derivatives
  • Nifedipine / metabolism
  • Nitrendipine
  • Rats
  • Rats, Inbred Strains
  • Verapamil / metabolism*

Substances

  • Ion Channels
  • Nitrendipine
  • Verapamil
  • Nifedipine
  • Calcium