Focused ultrasound delivery of Raman nanoparticles across the blood-brain barrier: potential for targeting experimental brain tumors

Nanomedicine. 2014 Jul;10(5):1075-87. doi: 10.1016/j.nano.2013.12.006. Epub 2013 Dec 27.

Abstract

Spectral mapping of nanoparticles with surface enhanced Raman scattering (SERS) capability in the near-infrared range is an emerging molecular imaging technique. We used magnetic resonance image-guided transcranial focused ultrasound (TcMRgFUS) to reversibly disrupt the blood-brain barrier (BBB) adjacent to brain tumor margins in rats. Glioma cells were found to internalize SERS capable nanoparticles of 50nm or 120nm physical diameter. Surface coating with anti-epidermal growth factor receptor antibody or non-specific human immunoglobulin G, resulted in enhanced cell uptake of nanoparticles in-vitro compared to nanoparticles with methyl terminated 12-unit polyethylene glycol surface. BBB disruption permitted the delivery of SERS capable spherical 50 or 120nm gold nanoparticles to the tumor margins. Thus, nanoparticles with SERS imaging capability can be delivered across the BBB non-invasively using TcMRgFUS and have the potential to be used as optical tracking agents at the invasive front of malignant brain tumors.

From the clinical editor: This study demonstrates the use of magnetic resonance image-guided transcranial focused ultrasound to open the BBB and enable spectral mapping of nanoparticles with surface enhanced Raman scattering (SERS)-based molecular imaging for experimental tumor tracking.

Keywords: Blood-brain barrier; Focused ultrasound; Giloma; Imaging; Nanoparticles.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / therapeutic use*
  • Blood-Brain Barrier / metabolism*
  • Blood-Brain Barrier / radiation effects*
  • Brain / metabolism
  • Brain Neoplasms / drug therapy*
  • Cell Line, Tumor
  • Drug Delivery Systems
  • ErbB Receptors / antagonists & inhibitors
  • Humans
  • Microscopy, Fluorescence
  • Nanoparticles / administration & dosage*
  • Nanoparticles / metabolism*
  • Rats
  • Sound*

Substances

  • Antineoplastic Agents
  • ErbB Receptors