Slow sodium channel inactivation in rat fast-twitch muscle

J Physiol. 1987 Feb:383:327-37. doi: 10.1113/jphysiol.1987.sp016411.

Abstract

1. Voltage-clamp Na+ currents (INa) were measured in rat fast-twitch fibres using the loose-patch-clamp technique. Changes in the conditioning membrane potential produced slow changes in the peak INa elicited by short test depolarizations, due to a slow inactivation process. 2. Inactivation was increased by application of steady depolarizing potentials and was reversed by steady hyperpolarizations. These changes in peak INa could be well fitted by single-exponential functions with time constants in the range of 1-4 min. 3. The steady-state values of the maximum peak INa at any potential could be well fitted by a function identical to the one describing the fast inactivation process. This gave a potential of -108 mV at which 50% of the channels were closed due to slow inactivation. 4. The maximum peak current densities obtained with the slow inactivation fully removed were as large as 20 mA cm-2.

MeSH terms

  • Animals
  • Female
  • Ion Channels / metabolism*
  • Male
  • Membrane Potentials
  • Muscles / physiology*
  • Rats
  • Rats, Inbred Strains
  • Sodium / metabolism*
  • Time Factors

Substances

  • Ion Channels
  • Sodium