Protective effects of exogenous β-hydroxybutyrate on paraquat toxicity in rat kidney

Biochem Biophys Res Commun. 2014 May 16;447(4):666-71. doi: 10.1016/j.bbrc.2014.04.074. Epub 2014 Apr 19.

Abstract

In this study, we demonstrated the protective effects of β-hydroxybutyrate (β-HB) against paraquat (PQ)-induced kidney injury and elucidated the underlying molecular mechanisms. By histological examination and renal dysfunction specific markers (serum BUN and creatinine) assay, β-HB could protect the PQ-induced kidney injury in rat. PQ-induced kidney injury is associated with oxidative stress, which was measured by increased lipid peroxidation (MDA) and decreased intracellular anti-oxidative abilities (SOD, CAT and GSH). β-HB pretreatment significantly attenuated that. Caspase-mediated apoptosis pathway contributed importantly to PQ toxicity, as revealed by the activation of caspase-9/-3, cleavage of PARP, and regulation of Bcl-2 and Bax, which were also effectively blocked by β-HB. Moreover, treatment of PQ strongly decreased the nuclear Nrf2 levels. However, pre-treatment with β-HB effectively suppressed this action of PQ. This may imply the important role of β-HB on Nrf2 pathway. Taken together, this study provides a novel finding that β-HB has a renoprotective ability against paraquat-induced kidney injury.

Keywords: Apoptosis; Kidney injury; Oxidative stress; Paraquat; β-Hydroxybutyrate.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3-Hydroxybutyric Acid / pharmacology*
  • Acute Kidney Injury / chemically induced
  • Acute Kidney Injury / metabolism
  • Acute Kidney Injury / prevention & control
  • Animals
  • Apoptosis / drug effects
  • Blood Urea Nitrogen
  • Caspase 3 / metabolism
  • Caspase 9 / metabolism
  • Catalase / metabolism
  • Creatinine / blood
  • Enzyme Activation / drug effects
  • Glutathione / metabolism
  • Herbicides / antagonists & inhibitors*
  • Herbicides / toxicity*
  • Kidney / drug effects*
  • Kidney / metabolism
  • Kidney / pathology
  • Lipid Peroxidation / drug effects
  • Male
  • NF-E2-Related Factor 2 / metabolism
  • Oxidative Stress / drug effects
  • Paraquat / antagonists & inhibitors*
  • Paraquat / toxicity*
  • Poly(ADP-ribose) Polymerases / metabolism
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • Rats
  • Rats, Wistar
  • Signal Transduction / drug effects
  • Superoxide Dismutase / metabolism
  • bcl-2-Associated X Protein / metabolism

Substances

  • Bax protein, rat
  • Herbicides
  • NF-E2-Related Factor 2
  • Nfe2l2 protein, rat
  • Proto-Oncogene Proteins c-bcl-2
  • bcl-2-Associated X Protein
  • Creatinine
  • Catalase
  • Superoxide Dismutase
  • Poly(ADP-ribose) Polymerases
  • Casp3 protein, rat
  • Casp9 protein, rat
  • Caspase 3
  • Caspase 9
  • Glutathione
  • Paraquat
  • 3-Hydroxybutyric Acid