Fucosylated chondroitin sulfate from sea cucumber improves insulin sensitivity via activation of PI3K/PKB pathway

J Food Sci. 2014 Jul;79(7):H1424-9. doi: 10.1111/1750-3841.12465.

Abstract

This study was to investigate the effects of fucosylated chondroitin sulfate (CHS) from sea cucumber on insulin sensitivity in skeletal muscle of type 2 diabetic mice induced by a high-fat high-sucrose diet (HFSD). CHS supplementation for 19 wk significantly improved insulin sensitivity by 20%, and reduced blood glucose and insulin levels. Western blotting assay showed that CHS significantly increased insulin-stimulated glucose transporter 4 (GLUT4) translocation to 1.7-fold, phosphorylation of phosphoinositide 3-kinase (PI3K) at p85 to 5.0-fold, protein kinase B (PKB) at Ser473 to 1.5-fold, and Thr308 to 1.6-fold in skeletal muscle. However, PI3K, PKB, and GLUT4 total proteins expression were unchangeable. In addition, qRT-PCR analysis proved that the insulin signaling was activated by CHS treatment, showing the increased mRNA expressions of glucose uptake-related key genes. It indicated that CHS improved insulin sensitivity by activation of PI3K/PKB signaling in skeletal muscle of type 2 diabetic mice. Identification of potential mechanism by which CHS increased insulin sensitivity might provide a new functional food or pharmaceutical application of sea cucumber.

Keywords: fucosylated chondroitin sulfate; insulin sensitivity; phosphoinositide 3-kinase; protein kinase B; sea cucumber.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Glucose
  • Chondroitin Sulfates / chemistry
  • Chondroitin Sulfates / pharmacology*
  • Diabetes Mellitus, Experimental / metabolism
  • Glucose Transporter Type 4 / metabolism
  • Hyperinsulinism
  • Insulin / blood
  • Insulin Resistance / physiology*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Muscle, Skeletal / metabolism
  • Phosphatidylinositol 3-Kinases / genetics
  • Phosphatidylinositol 3-Kinases / metabolism*
  • Phosphorylation / drug effects
  • Proto-Oncogene Proteins c-akt / genetics
  • Proto-Oncogene Proteins c-akt / metabolism*
  • Sea Cucumbers*
  • Signal Transduction / drug effects

Substances

  • Blood Glucose
  • Glucose Transporter Type 4
  • Insulin
  • fucosylated chondroitin sulfate
  • Chondroitin Sulfates
  • Phosphatidylinositol 3-Kinases
  • Proto-Oncogene Proteins c-akt