Biochemical characterization of soluble phospholipase A2 from rheumatoid synovial fluid

Agents Actions. 1989 Jun;27(3-4):477-80. doi: 10.1007/BF01972857.

Abstract

Radiolabeled E. coli, Phosphatidylethanolamine (PE) and Phosphatidylcholine (PC), were used to characterize the phospholipase A2 (PLA2) activity in synovial fluid (SF) from rheumatoid arthritis (RA) patients. Cell-free fractions of SF contain a PLA2 enzyme that preferentially releases [14C]oleic acid from E. coli, requires calcium and is optimally active at neutral pH. Purified PE, but not PC is also readily degraded by the soluble enzyme. A cell-associated PLA2 present in sonicates of SF mononuclear cells and neutrophils preferentially releases [3H]AA from E. coli. These studies suggest the presence of at least two different enzymes with activity of PLA2 in rheumatoid SF.

MeSH terms

  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology
  • Arthritis, Rheumatoid / enzymology*
  • Calcium / pharmacology
  • Edetic Acid / pharmacology
  • Escherichia coli / metabolism
  • Humans
  • Hydrogen-Ion Concentration
  • Micelles
  • Phosphatidylcholines / metabolism
  • Phosphatidylethanolamines / metabolism
  • Phospholipases / metabolism*
  • Phospholipases A / metabolism*
  • Phospholipases A2
  • Phospholipids / metabolism
  • Substrate Specificity
  • Synovial Fluid / enzymology*

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Micelles
  • Phosphatidylcholines
  • Phosphatidylethanolamines
  • Phospholipids
  • Edetic Acid
  • Phospholipases
  • Phospholipases A
  • Phospholipases A2
  • Calcium