Gut-liver axis improves with meloxicam treatment after cirrhotic liver resection

World J Gastroenterol. 2014 Oct 28;20(40):14841-54. doi: 10.3748/wjg.v20.i40.14841.

Abstract

Aim: To investigate the effect of meloxicam on the gut-liver axis after cirrhotic liver resection.

Methods: Forty-four male Wistar rats were assigned to three groups: (1) control group (CG); (2) bile duct ligation with meloxicam treatment (BDL + M); and (3) bile duct ligation without meloxicam treatment (BDL). Secondary biliary liver cirrhosis was induced via ligature of the bile duct in the BDL + M and BDL groups. After 2 wk, the animals underwent a 50% hepatectomy. In the BDL + M group 15 min prior to the hepatectomy, one single dose of meloxicam was administered. Parameters measured included: microcirculation of the liver and small bowel; portal venous flow (PVF); gastrointestinal (GI) transit; alanine aminotransferase (ALT); malondialdehyde; interleukin 6 (IL-6), transforming growth factor beta 1 (TGF-β1) and hypoxia-inducible factor 1 alpha (HIF-1α) levels; mRNA expression of cyclooxigenase-2 (COX-2), IL-6 and TGF-β1; liver and small bowel histology; immunohistochemical evaluation of hepatocyte and enterocyte proliferation with Ki-67 and COX-2 liver expression.

Results: Proliferative activity of hepatocytes after liver resection, liver flow and PVF were significantly higher in CG vs BDL + M and CG vs BDL group (P < 0.05), whereas one single dose of meloxicam ameliorated liver flow and proliferative activity of hepatocytes in BDL + M vs BDL group. COX-2 liver expression at 24 h observation time (OT), IL-6 concentration and mRNA IL-6 expression in the liver especially at 3 h OT, were significantly higher in BDL group when compared with the BDL + M and CG groups (P < 0.01, P < 0.001, P < 0.01, respectively). Liver and small bowel histology, according to a semi quantitative scoring system, showed better integrity in BDL + M and CG as compared to BDL group. ALT release and HIF-1α levels at 1 h OT were significantly higher in BDL + M compared to CG and BDL group (P < 0.001 and P < 0.01, respectively). Moreover, ALT release levels at 3 and 24 h OT were significantly higher in BDL group compared to CG, P < 0.01. GI transit, enterocyte proliferative activity and number of goblet cells were in favor of meloxicam treatment vs BDL group (P < 0.05, P < 0.001, P < 0.01, respectively). Additionally, villus length were higher in BDL + M as compared to BDL group.

Conclusion: One single dose of meloxicam administered after cirrhotic liver resection was able to cause better function and integrity of the remaining liver and small bowel.

Keywords: Cyclooxigenase-2; Gut-liver axis; Liver cirrhosis; Liver resection; Meloxicam; Microcirculation.

MeSH terms

  • Alanine Transaminase / blood
  • Animals
  • Cell Proliferation / drug effects
  • Cyclooxygenase 2 / genetics
  • Cyclooxygenase 2 / metabolism
  • Cyclooxygenase 2 Inhibitors / pharmacology*
  • Enterocytes / drug effects
  • Enterocytes / metabolism
  • Enterocytes / pathology
  • Gastrointestinal Transit / drug effects
  • Gene Expression Regulation
  • Hepatectomy*
  • Hepatocytes / drug effects
  • Hepatocytes / metabolism
  • Hepatocytes / pathology
  • Hypoxia-Inducible Factor 1, alpha Subunit / genetics
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Interleukin-6 / genetics
  • Interleukin-6 / metabolism
  • Intestine, Small / blood supply
  • Intestine, Small / drug effects*
  • Intestine, Small / metabolism
  • Intestine, Small / pathology
  • Intestine, Small / physiopathology
  • Lipid Peroxidation / drug effects
  • Liver / blood supply
  • Liver / drug effects*
  • Liver / metabolism
  • Liver / pathology
  • Liver / physiopathology
  • Liver / surgery*
  • Liver Circulation / drug effects
  • Liver Cirrhosis / diagnosis
  • Liver Cirrhosis / genetics
  • Liver Cirrhosis / metabolism
  • Liver Cirrhosis / physiopathology
  • Liver Cirrhosis / therapy*
  • Liver Regeneration / drug effects
  • Male
  • Malondialdehyde / blood
  • Meloxicam
  • Microcirculation / drug effects
  • RNA, Messenger / metabolism
  • Rats, Wistar
  • Thiazines / pharmacology*
  • Thiazoles / pharmacology*
  • Time Factors
  • Transforming Growth Factor beta1 / genetics
  • Transforming Growth Factor beta1 / metabolism

Substances

  • Cyclooxygenase 2 Inhibitors
  • Hif1a protein, rat
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Interleukin-6
  • RNA, Messenger
  • Tgfb1 protein, rat
  • Thiazines
  • Thiazoles
  • Transforming Growth Factor beta1
  • Malondialdehyde
  • Cyclooxygenase 2
  • Ptgs2 protein, rat
  • Alanine Transaminase
  • Meloxicam