Analysis of the kinetic mechanism of the bovine liver mitochondrial dihydroorotate dehydrogenase

Biochemistry. 1989 Feb 7;28(3):1222-6. doi: 10.1021/bi00429a040.

Abstract

The steady-state kinetic mechanism of highly purified bovine liver mitochondrial dihydroorotate dehydrogenase has been investigated. Initial velocity analysis using S-dihydroorotate and coenzyme Q6 revealed parallel-line, double-reciprocal plots, indicative of a ping-pong mechanism. The dead-end inhibition pattern with barbituric acid and the reactions with alternate cosubstrates methyl-S-dihydroorotate and menadione also point to a ping-pong mechanism. However, product orotate was found to be competitive with dihydroorotate and uncompetitive with Q6. These findings suggest that dihydroorotate dehydrogenase may follow a nonclassical, two-site ping-pong mechanism, typical of an enzyme that contains two non-overlapping and kinetically isolated substrate binding sites. That these two sites communicate by an intramolecular electron-transfer system involving FMN and perhaps an iron-sulfur center is also suggested by the kinetic behavior of the enzyme.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Binding, Competitive
  • Cattle
  • Dihydroorotate Oxidase / metabolism*
  • Kinetics
  • Mathematics
  • Mitochondria, Liver / enzymology*
  • Models, Theoretical
  • Oxidoreductases / metabolism*

Substances

  • Oxidoreductases
  • Dihydroorotate Oxidase