Dexamethasone but not the equivalent doses of hydrocortisone induces neurotoxicity in neonatal rat brain

Pediatr Res. 2015 May;77(5):618-24. doi: 10.1038/pr.2015.19. Epub 2015 Feb 9.

Abstract

Background: The use of dexamethasone (Dex) in premature infants to treat or prevent chronic lung disease adversely affects neurodevelopment. Recent clinical studies suggest that hydrocortisone (HC) is a safer alternative to Dex. We compared the effects of Dex and HC on neurotoxicity in newborn rats.

Methods: Rat pups of a neurodevelopmental stage equivalent to premature human neonates were administered Dex or HC either as a single dose on postnatal day (PD) 6, repeated doses on PD 4 to 6 or tapering doses at PD 3 to 6 by i.p. injection. Brain weight, caspase-3 activity, and apoptotic cells were measured at PD 7; learning capability, memory, and motor function were measured at juvenile age.

Results: Dex decreased both body and brain weight gain, while HC did not. Tapering and repeated doses of Dex increased caspase-3 activity, cleaved caspase-3 and terminal deoxynucleotidyl transferase dUTP nick end labeling (TUNEL)-positive cells but HC, except at high doses, did not. Dex impaired learning and memory capability at juvenile age, while the rats exposed to HC showed normal cognitive behavior.

Conclusion: HC is probably safer to use than Dex in the immediate postnatal period in neonatal rats. Cautious extrapolation of these findings to human premature infants is required.

MeSH terms

  • Animals
  • Animals, Newborn
  • Apoptosis
  • Brain / drug effects
  • Brain / physiopathology*
  • Caspase 3 / metabolism
  • Cognition / drug effects
  • Dexamethasone / administration & dosage
  • Dexamethasone / adverse effects*
  • Female
  • Hydrocortisone / administration & dosage
  • Hydrocortisone / adverse effects*
  • Learning / drug effects
  • Male
  • Memory / drug effects
  • Motor Skills / drug effects
  • Neurotoxicity Syndromes / pathology
  • Organ Size
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Dexamethasone
  • Casp3 protein, rat
  • Caspase 3
  • Hydrocortisone