Essential Roles of Intracellular Calcium Release Channels in Muscle, Brain, Metabolism, and Aging

Curr Mol Pharmacol. 2015;8(2):206-22. doi: 10.2174/1874467208666150507105105.

Abstract

Calcium (Ca(2+)) release from intracellular stores controls numerous cellular processes, including cardiac and skeletal muscle contraction, synaptic transmission and metabolism. The ryanodine receptors (RyRs: RyR1, RyR2, RyR3) and inositol 1,4,5-trisphosphate receptors (IP3Rs: IP3R1, IP3R2, IP3R3) are the major Ca(2+) release channels (CRCs) on the endo/sarcoplasmic reticulum (ER/SR). RyRs and IP3Rs comprise macromolecular signaling complexes that include modulatory proteins which regulate channel activity in response to extracellular signals resulting in intracellular Ca(2+) release. Here we focus on the roles of CRCs in heart, skeletal muscle, brain, metabolism, and aging.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Aging / physiology*
  • Brain / metabolism
  • Brain / pathology
  • Brain / physiopathology*
  • Energy Metabolism / physiology*
  • Humans
  • Inositol 1,4,5-Trisphosphate Receptors / metabolism
  • Inositol 1,4,5-Trisphosphate Receptors / physiology*
  • Intracellular Space / metabolism
  • Muscle, Skeletal / metabolism
  • Muscle, Skeletal / pathology
  • Muscle, Skeletal / physiopathology*
  • Protein Isoforms / metabolism
  • Protein Isoforms / physiology
  • Ryanodine Receptor Calcium Release Channel / metabolism
  • Ryanodine Receptor Calcium Release Channel / physiology*
  • Sarcoplasmic Reticulum / metabolism

Substances

  • Inositol 1,4,5-Trisphosphate Receptors
  • Protein Isoforms
  • Ryanodine Receptor Calcium Release Channel