Pacritinib Bests Available Therapies for Myelofibrosis

Cancer Discov. 2015 Jul;5(7):OF7. doi: 10.1158/2159-8290.CD-NB2015-080. Epub 2015 Jun 1.
No abstract available

MeSH terms

  • Blood Platelets / drug effects
  • Bridged-Ring Compounds / pharmacology
  • Bridged-Ring Compounds / therapeutic use*
  • Clinical Trials, Phase III as Topic
  • Humans
  • Janus Kinases / antagonists & inhibitors
  • Primary Myelofibrosis / drug therapy*
  • Primary Myelofibrosis / pathology
  • Pyrimidines / pharmacology
  • Pyrimidines / therapeutic use*
  • Spleen / drug effects

Substances

  • 11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-5,7,26-triazatetracyclo(19.3.1.1(2,6).1(8,12))heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene
  • Bridged-Ring Compounds
  • Pyrimidines
  • Janus Kinases