Rational drug design: Tuning kinase inhibitor residence time

Nat Rev Drug Discov. 2015 Jul;14(7):457. doi: 10.1038/nrd4673. Epub 2015 Jun 19.
No abstract available

Publication types

  • Comment

MeSH terms

  • Acrylamides / pharmacokinetics*
  • Animals
  • B-Lymphocytes / drug effects*
  • Cyanoacrylates / pharmacokinetics*
  • Female
  • Humans
  • Protein Kinase Inhibitors / pharmacokinetics*
  • Protein-Tyrosine Kinases / antagonists & inhibitors*

Substances

  • Acrylamides
  • Cyanoacrylates
  • Protein Kinase Inhibitors
  • Protein-Tyrosine Kinases