Clopidogrel Resistance after Minor Ischemic Stroke or Transient Ischemic Attack is Associated with Radiological Cerebral Small-Vessel Disease

J Stroke Cerebrovasc Dis. 2015 Oct;24(10):2348-57. doi: 10.1016/j.jstrokecerebrovasdis.2015.06.024. Epub 2015 Aug 21.

Abstract

Background: The objective of this study was to compare nonresponders (NR) and responders (R) to clopidogrel with respect to presence of microvascular and macrovascular pathology in a cohort of patients with recent minor ischemic stroke (IS) or transient ischemic attack (TIA).

Methods: Seventy-two patients treated with clopidogrel after IS or TIA were evaluated 1 month after onset. Platelet aggregation was measured by multiple electrode aggregometry (Multiplate). Nonresponse was defined according to recent consensus. The degree of cerebral small-vessel disease (cSVD) was evaluated on computed tomography scans of the brain using Fazekas scale for white matter changes. Carotid atherosclerosis was evaluated by ultrasound or computed tomography/magnetic resonance angiography.

Results: Twenty-two percent of patients were NR. Moderate to extensive cSVD was more common for NR than R, 56% versus 25%, odds ratio 3.9 (1.2-12), P = .03. Correspondingly, 39% of patients with cSVD were NR versus 14% of patients with no or mild cSVD. No differences were found between NR and R in prevalence or severity of carotid atherosclerosis. NR had higher platelet aggregation response than R after stimulation with arachidonic acid or thrombin receptor-activating peptide, indicating a general platelet hyperreactivity. In a univariate analysis, hypertension, previous IS, glucose intolerance, pulse pressure above median, and presence of moderate to extensive cSVD were associated with the NR phenotype.

Conclusions: Nonresponsiveness to clopidogrel after minor IS or TIA is associated with radiological cSVD but not with carotid atherosclerosis.

Practice/implications: Measurement of platelet function is warranted in patients with cSVD. Larger studies on alternative or tailored antiplatelet treatment for these patients should be initiated.

Keywords: Clopidogrel resistance; TIA; cerebral small-vessel disease; hypertension; ischemic stroke.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Blood Glucose
  • Carotid Artery Diseases
  • Cerebral Small Vessel Diseases / diagnosis
  • Cerebral Small Vessel Diseases / diagnostic imaging*
  • Clopidogrel
  • Cohort Studies
  • Female
  • Glomerular Filtration Rate
  • Humans
  • Ischemic Attack, Transient / drug therapy
  • Ischemic Attack, Transient / metabolism*
  • Male
  • Middle Aged
  • Neuroimaging
  • Platelet Aggregation
  • Platelet Aggregation Inhibitors / adverse effects*
  • Radiography
  • Statistics, Nonparametric
  • Stroke / drug therapy*
  • Stroke / metabolism*
  • Sweden
  • Ticlopidine / adverse effects
  • Ticlopidine / analogs & derivatives*
  • Ultrasonography

Substances

  • Blood Glucose
  • Platelet Aggregation Inhibitors
  • Clopidogrel
  • Ticlopidine