The multiple sclerosis-associated regulatory variant rs10877013 affects expression of CYP27B1 and VDR under inflammatory or vitamin D stimuli

Mult Scler. 2016 Jul;22(8):999-1006. doi: 10.1177/1352458515610208. Epub 2015 Oct 14.

Abstract

Background: Vitamin D deficit is considered an important risk factor for many inflammatory and autoimmune diseases.

Objective: To investigate the influence of the multiple sclerosis (MS)-associated regulatory variant rs10877013 on the expression of genes involved in vitamin D activation (CYP27B1), vitamin D receptor (VDR), and vitamin D degradation (CYP24A1) under inflammatory environment or vitamin D.

Methods: We used lipopolysaccharide and interferon-gamma (LPS+IFNγ) activated monocytes from 119 individuals and vitamin D-stimulated lymphoblastoid cell lines (LCLs, n = 109) of 1000 genomes to quantify the mRNA expression of vitamin D genes by quantitative reverse transcription polymerase chain reaction (RT-qPCR).

Results: We found that CYP27B1 mRNA expression level was associated with the rs10877013 genotypes (p = 5.0E-6) in LPS+IFNγ treated monocytes, but not in vitamin D-stimulated LCLs. Inversely, rs10877013 genotypes were associated with VDR expression in LCLs (p = 6.0E-4) but not in monocytes. Finally, CYP24A1 was highly induced by the active form of vitamin D and its expression correlated with the expression of VDR in LCLs but neither the MS-associated variant in the region (rs2248359) nor any other variant located in 1 Mb around CYP24A1 was associated with its expression.

Conclusions: The MS-associated variant rs10877013 is a genetic determinant that affects the functioning of the vitamin D system linking environmental and genetic factors.

Keywords: CYP24A1; CYP27B1; VDR; Vitamin D; functional variant rs10877013; gene expression regulation.

MeSH terms

  • 25-Hydroxyvitamin D3 1-alpha-Hydroxylase / genetics*
  • 25-Hydroxyvitamin D3 1-alpha-Hydroxylase / metabolism
  • Cell Line
  • Gene Expression Regulation
  • Humans
  • Interferon-gamma / pharmacology*
  • Lipopolysaccharides / pharmacology*
  • Monocytes / drug effects*
  • Monocytes / enzymology
  • Monocytes / immunology
  • Multiple Sclerosis / diagnosis
  • Multiple Sclerosis / enzymology
  • Multiple Sclerosis / genetics*
  • Multiple Sclerosis / immunology
  • Polymorphism, Single Nucleotide*
  • Receptors, Calcitriol / agonists
  • Receptors, Calcitriol / genetics*
  • Receptors, Calcitriol / metabolism
  • Time Factors
  • Vitamin D / pharmacology*
  • Vitamin D3 24-Hydroxylase / genetics
  • Vitamin D3 24-Hydroxylase / metabolism

Substances

  • Lipopolysaccharides
  • Receptors, Calcitriol
  • VDR protein, human
  • Vitamin D
  • Interferon-gamma
  • CYP24A1 protein, human
  • Vitamin D3 24-Hydroxylase
  • 25-Hydroxyvitamin D3 1-alpha-Hydroxylase
  • CYP27B1 protein, human