Human leukocyte and porcine pancreatic elastase: X-ray crystal structures, mechanism, substrate specificity, and mechanism-based inhibitors

Biochemistry. 1989 Mar 7;28(5):1951-63. doi: 10.1021/bi00431a001.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Catalysis
  • Humans
  • Leukocytes / enzymology*
  • Models, Biological
  • Molecular Sequence Data
  • Pancreas / enzymology*
  • Pancreatic Elastase / antagonists & inhibitors
  • Pancreatic Elastase / metabolism*
  • Protease Inhibitors / pharmacology
  • Protein Conformation
  • Structure-Activity Relationship
  • Substrate Specificity
  • Swine
  • X-Ray Diffraction

Substances

  • Protease Inhibitors
  • Pancreatic Elastase