Mechanism of Action and Applications of Interleukin 24 in Immunotherapy

Int J Mol Sci. 2016 Jun 2;17(6):869. doi: 10.3390/ijms17060869.

Abstract

Interleukin 24 (IL-24) is an important pleiotropic immunoregulatory cytokine, whose gene is located in human chromosome 1q32-33. IL-24's signaling pathways have diverse biological functions related to cell differentiation, proliferation, development, apoptosis, and inflammation, placing it at the center of an active area of research. IL-24 is well known for its apoptotic effect in cancer cells while having no such effect on normal cells. IL-24 can also be secreted by both immune and non-immune cells. Downstream effects of IL-24, after binding to the IL-20 receptor, can occur dependently or independently of the JAK/STAT signal transduction pathway, which is classically involved in cytokine-mediated activities. After exogenous addition of IL-24, apoptosis is induced in tumor cells independently of the JAK/STAT pathway. We have shown that IL-24 binds to Sigma 1 Receptor and this event induces endoplasmic reticulum stress, calcium mobilization, reactive oxygen species generation, p38MAPK activity, and ceramide production. Here we review IL-24's role in autoimmunity, infectious disease response, wound repair, and vascular disease. Detailed understanding of the pleiotropic roles of IL-24 signaling can assist in the selection of more accurate therapeutic approaches, as well as targeting of appropriate cell types in treatment strategy development, and ultimately achieve desired therapeutic effects.

Keywords: IL-24; Sigma 1 Receptor; cancer; endoplasmic reticulum (ER) stress; inflammatory disease.

Publication types

  • Review

MeSH terms

  • Animals
  • Cardiovascular Diseases / genetics
  • Cardiovascular Diseases / immunology
  • Cardiovascular Diseases / metabolism
  • Cardiovascular Diseases / therapy
  • Disease Resistance / genetics
  • Disease Resistance / immunology
  • Gene Expression
  • Humans
  • Immune System / cytology
  • Immune System / immunology
  • Immune System / metabolism
  • Immunity, Innate
  • Immunotherapy* / methods
  • Inflammation / genetics
  • Inflammation / immunology
  • Inflammation / metabolism
  • Inflammation / therapy
  • Interleukins / chemistry
  • Interleukins / genetics
  • Interleukins / metabolism*
  • Neoplasm Metastasis
  • Neoplasms / genetics
  • Neoplasms / immunology
  • Neoplasms / metabolism
  • Neoplasms / therapy
  • Neovascularization, Physiologic / genetics
  • Protein Binding
  • Receptors, Interleukin / metabolism
  • Signal Transduction
  • Wound Healing / genetics
  • Wound Healing / immunology

Substances

  • Interleukins
  • Receptors, Interleukin
  • interleukin-20 receptor
  • interleukin-24