EFFECT OF ε-AMINOCAPROIC ACID ON FIBRINOLYSIS IN PLASMA OF ASIAN ELEPHANTS (ELEPHAS MAXIMUS)

J Zoo Wildl Med. 2016 Jun;47(2):397-404. doi: 10.1638/2015-0255.1.

Abstract

ε-Aminocaproic acid (EACA) is a lysine analogue antifibrinolytic drug used to treat bleeding disorders in humans and domestic animals. Use in zoological medicine is rare and dose recommendations are anecdotal, but EACA may be a valuable therapeutic option for bleeding disorders in exotic species, including Asian elephants ( Elephas maximus ). This study used an in vitro model of hyperfibrinolysis and a thromboelastograph-based assay to estimate the therapeutic plasma concentration of EACA in Asian elephants (61.5 μg/ml, 95% CI = 34.6-88.5 μg/ml). Substantial but incomplete inhibition of lysis was seen at relatively low concentrations of EACA (40 μg/ml). Asian elephants appear sensitive to EACA-mediated inhibition of hyperfibrinolysis. Doses published for domestic animals, targeting higher plasma concentrations, may be inappropriate in this species.

Keywords: Asian elephant; Elephas maximus; fibrinolysis; thromboelastography; ε-aminocaproic acid.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminocaproic Acid / pharmacology*
  • Animals
  • Antifibrinolytic Agents / pharmacology*
  • Dose-Response Relationship, Drug
  • Elephants / blood*
  • Female
  • Fibrinolysis / drug effects*
  • Male
  • Thrombelastography / veterinary

Substances

  • Antifibrinolytic Agents
  • Aminocaproic Acid