C-phycocyanin suppresses transforming growth factor-β1-induced epithelial mesenchymal transition in human epithelial cells

Pharmacol Rep. 2017 Jun;69(3):426-431. doi: 10.1016/j.pharep.2016.12.013. Epub 2017 Jan 5.

Abstract

Background: Epithelial mesenchymal transition (EMT) is a process through which epithelial cells undergo multiple biochemical changes, causing them to differentiate into a mesenchymal-cell phenotype. This process has been shown to contribute to the development of fibrotic diseases. C-phycocyanin (C-PC) is a phycobiliprotein extracted from Spirulina platensis. This study was done to investigate the effect of C-PC on transforming growth factor-β1 (TGF-β1)-induced EMT and an EMT associated proliferation in human epithelial cell lines.

Methods: Human adenocarcinoma cell line, A549 and breast cancer cell line, MCF-7 were treated with TGF-β1, and EMT-related genes expression, cell proliferation and cell cycle arrest were examined.

Results: C-PC suppressed the EMT as assessed by reduced expression of vimentin, type-1-collagen and fibronectin, and increased E-cadherin expression in TGF-β1 treated cells. Further, TGF-β1 treatment induced cell cycle arrest in S and G2/M phase in A549 cells. However, TGF-β1-mediated cell cycle arrest was significantly reversed by combined treatment with C-PC.

Conclusions: The overall data suggested that C-PC suppresses TGF- β1-induced EMT and warrants further in vivo studies for future evaluation of C-PC as a potential antifibrotic agent.

Keywords: C-phycocyanin; Cell proliferation; Epithelial cells; Epithelial-to-mesenchymal transition; TGF-β1.

MeSH terms

  • A549 Cells
  • Adenocarcinoma / metabolism
  • Breast Neoplasms / metabolism
  • Cell Cycle Checkpoints / drug effects
  • Cell Proliferation / drug effects*
  • Epithelial Cells / drug effects*
  • Epithelial Cells / metabolism
  • Epithelial-Mesenchymal Transition / drug effects*
  • Female
  • Gene Expression Regulation / drug effects
  • Humans
  • MCF-7 Cells
  • Phycocyanin / isolation & purification
  • Phycocyanin / pharmacology*
  • Transforming Growth Factor beta1 / administration & dosage

Substances

  • Transforming Growth Factor beta1
  • Phycocyanin