Are there superagonists for calcium-activated potassium channels?

Channels (Austin). 2017 Nov 2;11(6):504-506. doi: 10.1080/19336950.2017.1376971. Epub 2017 Oct 5.
No abstract available

Keywords: EBIO; KCa2.2; KCa3.1; NS309; SKA-121; SKA-31; gating modulator; intermediate-conductance Ca2+-activated K+ channel; small-conductance Ca2+-activated K+ channel.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Binding Sites
  • Calcium / metabolism*
  • Calmodulin / metabolism*
  • Humans
  • Potassium Channels, Calcium-Activated / agonists*
  • Protein Binding
  • Protein Conformation

Substances

  • Calmodulin
  • Potassium Channels, Calcium-Activated
  • Calcium