Anti-inflammatory effects of Ginkgo biloba extract against trimethyltin-induced hippocampal neuronal injury

Inflammopharmacology. 2018 Feb;26(1):87-104. doi: 10.1007/s10787-017-0396-2. Epub 2017 Sep 16.

Abstract

Background: Despite the immense neuromodulatory potentials of Ginkgo biloba extract as a memory enhancer, its underlying mechanism seems inadequate particularly with regard to its anti-inflammatory properties.

Aim: The objective of the present study is to investigate the protective potentials of Ginkgo biloba extract (GBE) against hippocampal neuronal injury induced by trimethyltin (TMT), a potent neurotoxicant.

Methods: Male SD rats were administered trimethyltin (8.5 mg kg-1 b.wt) single intraperitoneal (i.p.) injection, followed by Ginkgo biloba extract (100 mg kg-1 b.wt i.p) for 21 days.

Results: The co-administration of GBE with TMT showed marked improvement in cognitive functions. Concomitantly, there was a significant decrease in oxidative stress as evident by reduction in MDA and total ROS levels. In addition, there was a marked suppression of astrocyte activation (GFAP), transcription factor NFκB and proinflammatory cytokines (TNF-α, IL-1α, 1L-6), which were found to be elevated by TMT administration. Histopathological observations showed remarkable improvement in hippocampal neuronal injury in the conjunctive group.

Conclusion: Therefore, it is suggested that Ginkgo biloba extract is an effective agent against trimethyltin-induced hippocampal neuronal loss owing to its antioxidative as well as anti-inflammatory properties.

Keywords: Cytokines; GFAP; Ginkgo biloba extract; Neuroinflammation; Proinflammatory; Trimethyltin.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology*
  • Antioxidants / metabolism
  • Cytokines / metabolism
  • Ginkgo Extract
  • Ginkgo biloba
  • Glial Fibrillary Acidic Protein / metabolism
  • Hippocampus / drug effects*
  • Hippocampus / metabolism
  • Inflammation / drug therapy*
  • Inflammation / metabolism
  • Male
  • Neurotoxicity Syndromes / drug therapy*
  • Neurotoxicity Syndromes / metabolism
  • Oxidative Stress / drug effects
  • Phytotherapy / methods
  • Plant Extracts / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Trimethyltin Compounds / pharmacology*
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Anti-Inflammatory Agents
  • Antioxidants
  • Cytokines
  • Glial Fibrillary Acidic Protein
  • Plant Extracts
  • Trimethyltin Compounds
  • Tumor Necrosis Factor-alpha
  • trimethyltin
  • Ginkgo biloba extract
  • Ginkgo Extract