Stereoselective Epimerizations of Glycosyl Thiols

Org Lett. 2017 Nov 3;19(21):5802-5805. doi: 10.1021/acs.orglett.7b02760.

Abstract

Glycosyl thiols are widely used in stereoselective S-glycoside synthesis. Their epimerization from 1,2-trans to 1,2-cis thiols (e.g., equatorial to axial epimerization in thioglucopyranose) was attained using TiCl4, while SnCl4 promoted their axial-to-equatorial epimerization. The method included application for stereoselective β-d-manno- and β-l-rhamnopyranosyl thiol formation. Complex formation explains the equatorial preference when using SnCl4, whereas TiCl4 can shift the equilibrium toward the 1,2-cis thiol via 1,3-oxathiolane formation.

Publication types

  • Research Support, Non-U.S. Gov't