[Phe8 psi(CH2-NH)Arg9]bradykinin, a B2 receptor selective agonist which is not broken down by either kininase I or kininase II

Eur J Pharmacol. 1988 Oct 11;155(1-2):193-5. doi: 10.1016/0014-2999(88)90423-2.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Pressure / drug effects
  • Bradykinin / analogs & derivatives*
  • Bradykinin / metabolism
  • Bradykinin / pharmacology
  • Carboxypeptidases / metabolism*
  • Dogs
  • In Vitro Techniques
  • Lysine Carboxypeptidase / metabolism*
  • Muscle, Smooth, Vascular / drug effects
  • Peptidyl-Dipeptidase A / metabolism*
  • Rabbits
  • Rats
  • Receptors, Bradykinin
  • Receptors, Neurotransmitter / drug effects*

Substances

  • Receptors, Bradykinin
  • Receptors, Neurotransmitter
  • bradykinin, Phe(8)-psi-CH2NH-Arg(9)-
  • Carboxypeptidases
  • Peptidyl-Dipeptidase A
  • Lysine Carboxypeptidase
  • Bradykinin