NR4A1 inhibition synergizes with ibrutinib in killing mantle cell lymphoma cells

Blood Cancer J. 2017 Nov 23;7(12):632. doi: 10.1038/s41408-017-0005-z.
No abstract available

Publication types

  • Letter
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adenine / analogs & derivatives
  • Antineoplastic Combined Chemotherapy Protocols / pharmacology*
  • Apoptosis / drug effects
  • Cell Line, Tumor
  • Drug Synergism
  • Humans
  • Lymphoma, Mantle-Cell / genetics*
  • Nuclear Receptor Subfamily 4, Group A, Member 1 / antagonists & inhibitors*
  • Oncogenes / genetics*
  • Piperidines
  • Pyrazoles / pharmacology
  • Pyrimidines / pharmacology

Substances

  • NR4A1 protein, human
  • Nuclear Receptor Subfamily 4, Group A, Member 1
  • Piperidines
  • Pyrazoles
  • Pyrimidines
  • ibrutinib
  • Adenine