Structure-binding-activity analysis of beta-adrenergic amines--I. Binding to the beta receptor and activation of adenylate cyclase

Biochem Pharmacol. 1978 May 15;27(10):1445-54. doi: 10.1016/0006-2952(78)90100-4.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenylyl Cyclases / metabolism*
  • Adrenergic beta-Agonists / metabolism
  • Adrenergic beta-Agonists / pharmacology*
  • Adrenergic beta-Antagonists / metabolism
  • Adrenergic beta-Antagonists / pharmacology*
  • Animals
  • Catecholamines / metabolism
  • Catecholamines / pharmacology
  • Enzyme Activation / drug effects
  • Erythrocyte Membrane / metabolism
  • Guanylyl Imidodiphosphate / pharmacology
  • In Vitro Techniques
  • Pindolol / analogs & derivatives
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, beta / metabolism*
  • Structure-Activity Relationship
  • Turkeys

Substances

  • Adrenergic beta-Agonists
  • Adrenergic beta-Antagonists
  • Catecholamines
  • Receptors, Adrenergic
  • Receptors, Adrenergic, beta
  • Guanylyl Imidodiphosphate
  • Pindolol
  • Adenylyl Cyclases