Cross-tolerance to the hypothermic effect of delta 8-tetrahydrocannabinol 11-hydroxy-delta 8-tetrahydrocannabinol and chlorpromazine in the mouse

Eur J Pharmacol. 1985 May 8;111(2):159-66. doi: 10.1016/0014-2999(85)90752-6.

Abstract

When a 5 mg/kg i.v. dose of delta 8-tetrahydrocannabinol (delta 8-THC) and 11-hydroxy-delta 8-tetrahydrocannabinol (11-OH-delta 8-THC) was administered daily to mice, tolerance to their hypothermic effects developed quickly. Cross-tolerance to the hypothermic effect also developed between delta 8-THC and 11-OH-delta 8-THC. Tolerance development was dose-dependent and dose-effect experiments indicated that the magnitude of the tolerance developed to 11-OH-delta 8-THC was greater than that to delta 8-THC. Both cannabinoids were cross-tolerant to chlorpromazine in the hypothermic effect, but not to morphine, pentobarbital and reserpine under the conditions used. The present results suggest that 11-OH-delta 8-THC has some role in the development of tolerance to the hypothermic effect of delta 8-THC in mice.

MeSH terms

  • Animals
  • Body Temperature / drug effects*
  • Chlorpromazine / pharmacology*
  • Dose-Response Relationship, Drug
  • Dronabinol / analogs & derivatives*
  • Dronabinol / pharmacology*
  • Drug Tolerance
  • Male
  • Mice
  • Mice, Inbred Strains
  • Morphine / pharmacology
  • Pentobarbital / pharmacology
  • Reserpine / pharmacology

Substances

  • 11-hydroxy-delta(8)-tetrahydrocannabinol
  • delta-8-tetrahydrocannabinol
  • Morphine
  • Dronabinol
  • Reserpine
  • Pentobarbital
  • Chlorpromazine