Thymosin fraction 5 re-evaluated after 35 years by high-resolution mass spectrometry

Expert Opin Biol Ther. 2018 Jul;18(sup1):199-203. doi: 10.1080/14712598.2018.1474196.

Abstract

Objectives: We reevaluated a lyophilized sample of thymosin fraction 5, stored for 37 years at room temperature, by high-resolution mass spectrometry in terms of stability and yet uncharacterized polypeptides that could be biological important substances.

Methods: A top-down proteomic platform based on high-performance liquid chromatography (HPLC) coupled to high-resolution LTQ-Orbitrap mass spectrometry (MS) was applied to molecular characterization of polypeptides present in thymosin fraction 5.

Results: We detected more than 100 monoisotopic masses corresponding to thymosin β4 and truncated forms of ubiquitin, prothymosin α, thymosin β4, and thymosin β9. Additionally, we discovered a new polypeptide present in thymosin fraction 5 and identified it as intact SH3 domain-binding glutamic acid-rich-like protein 3.

Conclusion: In spite of the well-known proteolytic processes inherent to the preparation of thymosin fraction 5, still uncharacterized polypeptides as well as truncated forms of already well-known thymosins are present in fraction 5 after long-term storage. Therefore, continuing characterization of thymosin fraction 5 is even nowadays highly promising.

Keywords: SH3 domain-binding; Top-down proteomics; glutamic acid-rich-like protein 3; thymosin fraction 5; α-Thymosins; β-Thymosins.

MeSH terms

  • Animals
  • Chromatography, High Pressure Liquid
  • Drug Stability
  • Drug Storage
  • Freeze Drying
  • Humans
  • Mass Spectrometry / methods*
  • Protein Precursors / analysis
  • Protein Precursors / isolation & purification
  • Proteomics / methods
  • Thymosin / analogs & derivatives*
  • Thymosin / analysis
  • Thymosin / chemistry
  • Thymosin / isolation & purification
  • Thymosin beta(4)
  • Time Factors
  • Ubiquitin / analysis
  • Ubiquitin / isolation & purification

Substances

  • Protein Precursors
  • Thymosin
  • Ubiquitin
  • Thymosin beta(4)
  • prothymosin alpha
  • thymosin fraction 5
  • thymosin beta(9)