Targeting MEK in vemurafenib-resistant hairy cell leukemia

Leukemia. 2019 Feb;33(2):541-545. doi: 10.1038/s41375-018-0270-2. Epub 2018 Oct 19.
No abstract available

Publication types

  • Case Reports
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Antineoplastic Agents / pharmacology
  • Azetidines / therapeutic use*
  • Drug Resistance, Neoplasm / drug effects*
  • Humans
  • Leukemia, Hairy Cell / drug therapy*
  • Leukemia, Hairy Cell / pathology
  • MAP Kinase Kinase 1 / antagonists & inhibitors*
  • MAP Kinase Kinase 1 / genetics
  • Male
  • Piperidines / therapeutic use*
  • Prognosis
  • Salvage Therapy*
  • Vemurafenib / pharmacology*

Substances

  • Antineoplastic Agents
  • Azetidines
  • Piperidines
  • Vemurafenib
  • MAP Kinase Kinase 1
  • MAP2K1 protein, human
  • cobimetinib