Decrease in glucokinase and glucose-6-phosphatase and increase in hexokinase in putative preneoplastic lesions of rat liver

J Cancer Res Clin Oncol. 1987;113(5):430-6. doi: 10.1007/BF00390036.

Abstract

Preneoplastic liver lesions were produced in female Wistar rats by oral administration of 2-acetylaminofluorene for 165 days succeeded by a carcinogen-free standard diet up to 420 days. During the treatment numerous altered hepatic foci (AHF) and hyperplastic nodules (HN) were detected histochemically by a focal decrease or lack of adenosine-5-triphosphatase and glucose-6-phosphatase (G-6-Pase) activities. In addition, the immunohistochemically demonstrable amount of L-type pyruvate kinase was clearly reduced. The histochemically demonstrated decrease of G-6-Pase was substantiated by microbiochemical determination of the enzyme activity in microdissected material. Moreover, during the experimental period a continuous decrease in glucokinase and an increase in hexokinase was detected microbiochemically within AHF and HN. These alterations indicate a shift in the carbohydrate metabolism from gluconeogenesis to glucose utilization and pentose-phosphate-pathway for biosynthesis of nucleic acids. Beside other oncofetal markers, HK may be used as indicator of the early stages of liver carcinogenesis.

MeSH terms

  • 2-Acetylaminofluorene
  • Adenosine Triphosphatases / metabolism
  • Animals
  • Female
  • Glucokinase / metabolism*
  • Glucose-6-Phosphatase / metabolism*
  • Hexokinase / metabolism*
  • Histocytochemistry
  • Liver Neoplasms / chemically induced
  • Liver Neoplasms / enzymology*
  • Precancerous Conditions / chemically induced
  • Precancerous Conditions / enzymology*
  • Rats
  • Rats, Inbred Strains

Substances

  • 2-Acetylaminofluorene
  • Hexokinase
  • Glucokinase
  • Glucose-6-Phosphatase
  • Adenosine Triphosphatases