Time dependent degeneration of the nigrostriatal tract in mice with 6-OHDA lesioned medial forebrain bundle and the effect of activin A on L-Dopa induced dyskinesia

BMC Neurosci. 2019 Feb 13;20(1):5. doi: 10.1186/s12868-019-0487-7.

Abstract

Background: Accurately assessing promising therapeutic interventions for human diseases depends, in part, on the reproducibility of preclinical disease models. With the development of transgenic mice, the rapid adaptation of a 6-OHDA mouse model of Parkinson's disease that was originally described for the use in rats has come with a lack of a comprehensive characterization of lesion progression. In this study we therefore first characterised the time course of neurodegeneration in the substantia nigra pars compacta and striatum over a 4 week period following 6-OHDA injection into the medial forebrain bundle of mice. We then utilised the model to assess the anti-dyskinetic efficacy of recombinant activin A, a putative neuroprotectant and anti-inflammatory that is endogenously upregulated during the course of Parkinson's disease.

Results: We found that degeneration of fibers in the striatum was fully established within 1 week following 6-OHDA administration, but that the loss of neurons continued to progress over time, becoming fully established 3 weeks after the 6-OHDA injection. In assessing the anti-dyskinetic efficacy of activin A using this model we found that treatment with activin A did not significantly reduce the severity, or delay the time-of-onset, of dyskinesia.

Conclusion: First, the current study concludes that a 3 week duration is required to establish a complete lesion of the nigrostriatal tract following 6-OHDA injection into the medial forebrain bundle of mice. Second, we found that activin A was not anti-dyskinetic in this model.

Keywords: Abnormal involuntary movements; Neuroinflammation; Parkinson’s disease; Stereology; Striatum; Substantia nigra pars compacta.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Activins / pharmacology*
  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology
  • Antiparkinson Agents / adverse effects
  • Antiparkinson Agents / pharmacology
  • Disease Progression
  • Dyskinesia, Drug-Induced / drug therapy*
  • Dyskinesia, Drug-Induced / pathology
  • Dyskinesia, Drug-Induced / physiopathology
  • Levodopa / adverse effects
  • Levodopa / pharmacology
  • Male
  • Medial Forebrain Bundle / drug effects
  • Medial Forebrain Bundle / pathology
  • Medial Forebrain Bundle / physiopathology*
  • Mice, Inbred C57BL
  • Neurodegenerative Diseases / drug therapy
  • Neurodegenerative Diseases / pathology
  • Neurodegenerative Diseases / physiopathology*
  • Neurons / drug effects
  • Neurons / pathology
  • Neurons / physiology
  • Neuroprotective Agents / pharmacology*
  • Oxidopamine
  • Parkinsonian Disorders / drug therapy*
  • Parkinsonian Disorders / pathology
  • Parkinsonian Disorders / physiopathology
  • Random Allocation
  • Treatment Failure

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Antiparkinson Agents
  • Neuroprotective Agents
  • activin A
  • Activins
  • Levodopa
  • Oxidopamine