Dissociation of the anorectic actions of 5-HTP and fenfluramine

Psychopharmacology (Berl). 1986;89(2):216-20. doi: 10.1007/BF00310632.

Abstract

The possible peripheral anorectic actions of 5-hydroxytryptophan (5-HTP) and fenfluramine were examined in food-deprived rats. In a 1-h feeding test the peripherally acting 5-HT antagonist, xylamidine, attenuated the reductions in food intake induced by 5-HT and 5-HTP but not fenfluramine. Thus, the anorectic action of 5-HTP appears to be mediated in part by peripheral 5-HT receptors. Microstructural analyses showed that 5-HTP and fenfluramine induced decreases in eating rate and bout size. Xylamidine reversed the effect of 5-HTP on eating rate, and induced a slight increase in bout size in its own right. Therefore, the peripheral effect of 5-HTP appears to be a slowing of eating rate. No effects of xylamidine on fenfluramine induced changes in feeding were observed. The results indicate a dissociation of the anorectic effects of 5-HTP and fenfluramine based on a peripheral action of 5-HTP. The peripheral action of 5-HTP differs from the previously reported reductions in bout size and bout duration induced by 5-HT. Possible mechanisms for this difference in the peripheral actions of 5-HT and 5-HTP are discussed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amidines / pharmacology
  • Animals
  • Anorexia / chemically induced
  • Appetite Depressants / pharmacology*
  • Eating / drug effects
  • Fenfluramine / pharmacology*
  • Male
  • Rats
  • Receptors, Serotonin / drug effects
  • Serotonin / pharmacology*
  • Serotonin / physiology
  • Serotonin Antagonists / pharmacology

Substances

  • Amidines
  • Appetite Depressants
  • Receptors, Serotonin
  • Serotonin Antagonists
  • Fenfluramine
  • Serotonin
  • xylamidine