Glycoprotein V hydrolysis by thrombin. Lack of correlation with secretion

Thromb Res. 1985 Jun 15;38(6):641-8. doi: 10.1016/0049-3848(85)90207-5.

Abstract

Platelet membrane glycoprotein V (GPV) was hydrolyzed during thrombin-induced platelet aggregation releasing a fragment GPVfl into the supernatant. Hydrolysis of GPV required catalytically active thrombin and was diminished by chemical modification of the fibrinogen binding site of thrombin. Half-maximal liberation of GPVfl occurred at a 10-fold higher concentration of thrombin than was required for half-maximal release. Time course studies at several thrombin concentrations showed disparate release of GPVfl and thrombospondin. These results emphasize the complexity of the initial events in thrombin-induced platelet activation.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Binding Sites
  • Blood Platelets / metabolism*
  • Chymotrypsin / metabolism
  • Cytoplasmic Granules / metabolism
  • Fibrinogen / metabolism
  • Glycoproteins / metabolism*
  • Humans
  • Hydrolysis
  • Membrane Proteins / metabolism*
  • Platelet Membrane Glycoproteins
  • Thrombin / metabolism*
  • Thrombospondins

Substances

  • Glycoproteins
  • Membrane Proteins
  • Platelet Membrane Glycoproteins
  • Thrombospondins
  • Fibrinogen
  • Chymotrypsin
  • Thrombin