Receptor-Interacting Protein Kinase 3 (RIPK3) inhibits autophagic flux during necroptosis in intestinal epithelial cells

FEBS Lett. 2020 May;594(10):1586-1595. doi: 10.1002/1873-3468.13748. Epub 2020 Feb 16.

Abstract

Autophagy is an intracellular process that regulates the degradation of cytosolic proteins and organelles. Dying cells often accumulate autophagosomes. However, the mechanisms by which necroptotic stimulation induces autophagosomes are not defined. Here, we demonstrate that the activation of necroptosis with TNF-α plus the cell-permeable pan-caspase inhibitor Z-VAD induces LC3-II and LC3 puncta, markers of autophagosomes, via the receptor-interacting protein kinase 3 (RIPK3) in intestinal epithelial cells. Surprisingly, necroptotic stimulation reduces autophagic activity, as evidenced by enlarged puncta of the autophagic substrate SQSTM1/p62 and its increased colocalization with LC3. However, necroptotic stimulation does not induce the lysosomal-associated membrane protein 1 (LAMP1) nor syntaxin 17, which mediates autophagosome-lysosome fusion, to colocalize with LC3. These data indicate that necroptosis attenuates autophagic flux before the lysosome fusion step. Our findings may provide insights into human diseases involving necroptosis.

Keywords: RIPK3; SQSTM1/p62; STX17; autophagy; necroptotic stimulation; necrostatin-1.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Autophagosomes / drug effects
  • Autophagosomes / metabolism
  • Autophagy* / drug effects
  • Cell Line, Tumor
  • Epithelial Cells / cytology*
  • Epithelial Cells / drug effects
  • Epithelial Cells / enzymology*
  • Epithelial Cells / metabolism
  • Humans
  • Intestines / cytology*
  • Lysosomes / drug effects
  • Lysosomes / metabolism
  • Microtubule-Associated Proteins / metabolism
  • Necroptosis* / drug effects
  • Oligopeptides / pharmacology
  • Receptor-Interacting Protein Serine-Threonine Kinases / metabolism*
  • Sequestosome-1 Protein / metabolism
  • Tumor Necrosis Factor-alpha / pharmacology

Substances

  • Microtubule-Associated Proteins
  • Oligopeptides
  • SQSTM1 protein, human
  • Sequestosome-1 Protein
  • Tumor Necrosis Factor-alpha
  • benzyloxycarbonyl-valyl-alanyl-aspartic acid
  • RIPK3 protein, human
  • Receptor-Interacting Protein Serine-Threonine Kinases