Different solid forms for optimizing route of administration of the herpes drug Pritelivir

Medchemcomm. 2019 Aug 9;10(11):1867-1870. doi: 10.1039/c9md00233b. eCollection 2019 Nov 1.

Abstract

Pritelivir (AIC316, BAY 57-1293) was discovered as a highly potent drug against herpes simplex viruses with a novel mode of action, i.e. inhibition of the viral helicase-primase. A side by side comparison of the oral form against Valtrex™ in patients with genital herpes, showed superiority in phase II testing for Pritelivir. A number of different solid forms have been generated for additional, e.g. systemic, or topical applications.

Publication types

  • Review