Emerging therapeutic targets for neuroblastoma

Expert Opin Ther Targets. 2020 Sep;24(9):899-914. doi: 10.1080/14728222.2020.1790528. Epub 2020 Oct 6.

Abstract

Introduction: Neuroblastoma (NB) is the prime cancer of infancy, and accounts for 9% of pediatric cancer deaths. While children diagnosed with clinically stable NB experience a complete cure, those with high-risk disease (HR-NB) do not recover, despite intensive therapeutic strategies. Development of novel and effective targeted therapies is needed to counter disease progression, and to benefit long-term survival of children with HR-NB.

Areas covered: Recent studies (2017-2020) pertinent to NB evolution are selectively reviewed to recognize novel and effective therapeutic targets. The prospective and promising therapeutic targets/strategies for HR-NB are categorized into (a) targeting oncogene-like and/or reinforcing tumor suppressor (TS)-like lncRNAs; (b) targeting oncogene-like microRNAs (miRs) and/or mimicking TS-miRs; (c) targets for immunotherapy; (d) targeting epithelial-to-mesenchymal transition and cancer stem cells; (e) novel and beneficial combination approaches; and (f) repurposing drugs and other strategies in development.

Expert opinion: It is highly unlikely that agents targeting a single candidate or signaling will be beneficial for an HR-NB cure. We must develop efficient drug deliverables for functional targets, which could be integrated and advance clinical therapy. Fittingly, the looming evidence indicated an aggressive evolution of promising novel and integrative targets, development of efficient drugs, and improvised strategies for HR-NB treatment.

Keywords: Emerging therapeutics; high-risk Neuroblastoma; immunotherapy; long non-coding RNAs; micro RNAs; novel combinations; novel drugs.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology*
  • Child
  • Disease Progression
  • Drug Development
  • Epithelial-Mesenchymal Transition / drug effects
  • Humans
  • Immunotherapy / methods
  • Infant
  • Molecular Targeted Therapy*
  • Neoplastic Stem Cells / metabolism
  • Neuroblastoma / drug therapy*
  • Neuroblastoma / pathology
  • Survival Rate

Substances

  • Antineoplastic Agents