Safety and tolerability of nabiximols oromucosal spray: a review of real-world experience in observational studies, registries, and case reports

Expert Rev Neurother. 2021 May;21(5):547-558. doi: 10.1080/14737175.2021.1904896. Epub 2021 Mar 30.

Abstract

Introduction: : Nabiximols oromucosal spray,a cannabis-based medicine containing a balanced ratio of Δ-9-tetrahydrocannabinol and cannabidiol, is approved widely as an add-on therapy for symptomatic relief of spasticity in people with multiple sclerosis (MS). Most safety data for nabiximols derive from use in MS spasticity, with some data available from the analgesia area.

Areas covered: : This review compiles safety and tolerability data from all published observational studies, registry analyses, and case reports identified in systematic searches in which nabiximols oromucosal spray was investigated for spasticity (n = 20) and/or chronic non-cancer pain (n = 4). Aligning with the known safety profile of nabiximols as demonstrated in randomized controlled trials, common adverse events reported consistently across studies conducted under clinical practice conditions were dizziness, fatigue and somnolence. The serious adverse event (SAE) rate with nabiximols in MS spasticityobservational studies was 3.1% (137/4351). A total of 39 treatment-related SAEs were reported in 32 patients with spasticity, all of which (where specified) were resolved. No treatment-related SAEs were recorded in nabiximols pain studies.

Expert opinion: : Real-world experience with nabiximols oromucosal spray in treating spasticity and chronic pain indicates that, overall, it is well tolerated and has a good safety profile.

Keywords: Nabiximols; multiple sclerosis spasticity; neurological pain; observational studies; safety; sativex; tolerability.

Publication types

  • Case Reports
  • Review

MeSH terms

  • Analgesics, Opioid
  • Cannabidiol* / therapeutic use
  • Chronic Pain*
  • Dronabinol / adverse effects
  • Drug Combinations
  • Humans
  • Multiple Sclerosis* / drug therapy
  • Muscle Spasticity / drug therapy
  • Registries

Substances

  • Analgesics, Opioid
  • Drug Combinations
  • Cannabidiol
  • Dronabinol
  • nabiximols