[Analgesic activity of derivatives of 7-amino-2,3-polymethylenindoles and their congeners]

Farmaco Sci. 1988 Feb;43(2):113-23.
[Article in Italian]

Abstract

Some N-trifluoromethylsulphonyl and N-trifluoroacetylderivatives of 7-amino-2,3-polymethyleneindoles and of 7-amino-3-propylindole [(I) - (XIII)] were prepared and tested, together with corresponding aniline derivates [(XIV) - (XIX)] and with N-trifluoromethylsulphonylcyclopentylamine (XX), against formic acid induced writhings in mice. With very few exceptions, at the oral dose of 0.167 mmole/kg, they proved from 2 to 3.4 times more active than acetanilide.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analgesics / chemical synthesis*
  • Analgesics / pharmacology
  • Aniline Compounds / chemical synthesis*
  • Aniline Compounds / pharmacology
  • Animals
  • Chemical Phenomena
  • Chemistry
  • Cyclopentanes / chemical synthesis
  • Cyclopentanes / pharmacology
  • Female
  • Indoles / chemical synthesis*
  • Indoles / pharmacology
  • Mice

Substances

  • Analgesics
  • Aniline Compounds
  • Cyclopentanes
  • Indoles