Expeditious synthesis and preliminary antimicrobial activity of deflazacort and its precursors

RSC Adv. 2019 Jul 10;9(37):21519-21524. doi: 10.1039/c9ra03673c. eCollection 2019 Jul 5.

Abstract

The synthesis of deflazacort (DFZ) and a preliminary evaluation of its microbial activity against the human pathogens Acinetobacter baumannii and Staphylococcus aureus is herein reported. While DFZ is inactive, one of its synthetic precursors showed a strong antibacterial activity against both Gram-negative and -positive bacteria.